Small Molecule Medicinal Chemistry: Strategies and by Werngard Czechtizky,Peter Hamley PDF

By Werngard Czechtizky,Peter Hamley

ISBN-10: 1118771605

ISBN-13: 9781118771600

Stressing strategic and technological strategies to medicinal chemistry demanding situations, this publication offers tools and practices for optimizing the chemical points of drug discovery. Chapters speak about advantages, demanding situations, case reports, and views for making improvements to drug discovery courses with admire to caliber and costs.

•    Focuses on small molecules and their severe position in medicinal chemistry, reviewing chemical and fiscal merits, demanding situations, and developments within the box from perspectives
•    Discusses novel techniques and key issues, like screening assortment enhancement, threat sharing, HTS triage, new lead discovering methods, diversity-oriented synthesis, peptidomimetics, typical items, and excessive throughput medicinal chemistry approaches
•    Explains find out how to lessen design-make-test cycle occasions through integrating medicinal chemistry, actual chemistry, and ADME profiling techniques
•    Includes descriptive case stories, examples, and purposes to demonstrate new applied sciences and supply step by step reasons to allow them in a laboratory setting

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Small Molecule Medicinal Chemistry: Strategies and Technologies by Werngard Czechtizky,Peter Hamley

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